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U 89843A
CAS No. 157013-32-6
U 89843A ( —— )
产品货号. M27731 CAS No. 157013-32-6
U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥7857 | 有现货 |
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| 50MG | ￥16038 | 有现货 |
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| 100MG | ￥20250 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称U 89843A
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.
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产品描述U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.(In Vitro):In the alpha 1 beta 2 gamma 2 subtype of GABAA receptors expressed in human embryonic kidney cells, U 89843A dose-dependently enhanced 5 microM GABA-induced Cl- currents with a maximal enhancement of 362 +/- 91%, a half-maximal concentration of 2 +/- 0.4 microM and a slope factor of 1.1 +/- 0.4. U 89843A also inhibited [35S]t-butylbicyclophosphorothionate binding in rat cerebrocortical membranes with a similar half-maximal inhibitory concentration.
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同义词——
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通路Others
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靶点Other Targets
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受体acetylcholinesterase
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研究领域——
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适应症——
化学信息
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CAS Number157013-32-6
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分子量321.9
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分子式C16H24ClN5
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纯度>98% (HPLC)
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溶解度——
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SMILESCl.Cc1cc2c(nc(nc2n1C)N1CCCC1)N1CCCC1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Dafforn A, et al. Acetylcholinesterase inhibition by the ketone transition state analog phenoxyacetone and 1-halo-3-phenoxy-2-propanones. Biochem Biophys Res Commun. 1982 Jan 29;104(2):597-602.
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